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Cn1nncc1CCNC(=O)C(CC1CC1)NC(=O)Cc1ccoc1 |
Cn1nncc1CN(Cc1c[nH]c2cnccc12)CC1CC(Cl)(Cl)C1 |
Cn1nncc1CN(Cc1cc2ncncc2s1)CC(O)C1(C)CC1 |
Cn1nnnc1C(c1cn2cc(F)ccc2n1)N1C[C@H]2C[C@@H]1CS2=O |
Cn1nnnc1C1(NC(C)(C(N)=O)c2ccccc2)CCC(=O)NC1 |
Cn1nnnc1C1(NCc2cc(F)cc(Cl)c2)CC[C@H]2CCC[C@H]2C1 |
Cn1nnnc1CNC(=O)C12CC(CO1)N(C(=O)[C@H]1CCC(=O)O1)C2 |
FC(F)(F)C(F)(F)Oc1cccc(-n2cc(COC3CNC3)nn2)c1 |
FC(F)(F)C1=CC=C(\C=C\C2=NC(COC3=CC=C(CCCCN4C=CN=N4)C=C3)=CO2)C=C1 |
FC(F)(F)CN1CCC(CNc2ncnc3ncn(C4CC4)c23)CC1 |
FC(F)(F)c1cc(CNC2(c3ncc4c(n3)CCC4)CC2)cc(Cl)n1 |
FC(F)(F)c1ccnc(CN(CCCOCC2CCC2)CC2CC2)c1 |
FC(F)C(F)(F)CNc1ncnc(N2CCC(OCC3CC3)CC2)n1 |
FC(F)OC1CCC(Nc2ccccc2OCC2CCCCO2)CC1 |
FC1=C(Cl)C=C(NC2=NC=NC3=CC(OCCCN4CCOCC4)=C(NC(=O)C=C)C=C23)C=C1 |
FC1=CCCN(c2nc3c(c(NCC[C@H]4C[C@@H]4C4CC4)n2)CSC3)C1 |
FCCCNc1nc(NCCOC2CCSCC2)c2ncccc2n1 |
FCCCn1nnnc1C1(N[C@@H]2CCC[C@H]2F)CC2CC=CCC2C1 |
Fc1cc(Cl)cc(CNc2nc(N3CCSCC3)c3sccc3n2)c1 |
Fc1cc(F)c(CN(CCC(F)(F)F)CC2CC3CCC2O3)cc1F |
Fc1ccc(Cl)c(CNc2cc(N3CC4COCC(C4)C3)ncn2)c1 |
Fc1ccc(NC2CNC(c3ccccc3)C2)cc1OCC(F)(F)F |
Fc1ccc(OC2CCN(Cc3cnn(CC(F)(F)F)c3)CC2)nc1 |
Fc1ccc(Oc2nc3ccccc3n3nnnc23)cc1OC(F)F |
Fc1ccc(SCCNCc2c(F)cccc2OCC(F)(F)F)cc1 |
Fc1ccc2nc(NCCOc3ccc(C(F)(F)F)nc3)ncc2c1 |
Fc1cccc(CNCc2ncc(C(F)(F)F)cc2Cl)c1OC(F)F |
Fc1cccc2c(C(NC3CCC3)c3nnnn3C3COC3)n[nH]c12 |
Fc1cccnc1CCN(Cc1cccs1)CC1CC2(C1)OCCO2 |
Fc1cnc(CNc2ccnc3c(OCC(F)F)cccc23)cc1Br |
N#CC(C(=O)C12CC(C#N)(C1)C2)c1nc2cc(C(F)(F)F)ccc2s1 |
N#CC1(C(=O)NC2CCCN(c3cccc(C(F)(F)F)c3)C2)CCC1 |
N#CC1(C(=O)NCC2(C(=O)NCC[C@H]3CCC(=O)N3)CC2)CC(=O)C1 |
N#CC1(C(=O)NCCC(=O)NC2CCOCC23CCC3)CC2CC2C1 |
N#CC1(C2CCCC2)CCN(S(=O)(=O)c2cnn(CC(F)F)c2)CC1 |
N#CC1(CC(=O)N2CCC(F)(CNC(=O)CCOC3CCC3)C2)CC1 |
N#CC1(CN(CCC2CC2(Cl)Cl)Cc2ccc([N+](=O)[O-])cn2)CCC1 |
N#CC1(F)CN(C(=O)C(CC2CC2)NC(=O)C2CC3CC(=O)C2O3)C1 |
N#CC1(F)CN(C(=O)C2(CNC(=O)C3CCCN3C3CC3)CCC2)C1 |
N#CC12CC(C(=O)NC(CNC(=O)c3cnc[nH]3)C3CCOC3)(C1)C2 |
N#CC12CCC(C(=O)N3CCCC3c3ccc(F)cc3F)(CC1)CC2 |
N#CC1=C(C(=O)NCc2cc(C(=O)Nn3cccn3)ccn2)CCC1 |
N#CC1CC2(CNC(=O)c3cc4cc5c(cc4[nH]3)OCCO5)CC1C2 |
N#CC1CCC(C(=O)N2CC3(CN(C(=O)c4cc(Cl)[nH]n4)C3)C2)CC1 |
N#CC1CCCN(C(=O)C(CC(F)F)NC(=O)C2=CC3C=CC2C3)C1 |
N#CC1CCCN(c2cc(N3CCCC4(CC=CCC4)C3)ncn2)C1 |
N#CC1CCN(c2nc(NCC3CC34CC4)nc3c(F)cccc23)C1 |
N#CCC1(C(=O)N(Cc2cn(C3CC3)cn2)CC2CCSCC2)CC1 |
N#CCCCC(Nc1ccc(O)cc1)c1nnnn1CCCC1CC1 |
N#CCCCCC(=O)N1C[C@H](O)C[C@@H]1C(=O)NCC1(F)CCCCC1 |
N#CCCCCC(=O)NCC1(NC(=O)c2ccc(=O)[nH]c2)CCCC1 |
N#CCCCCCC(=O)NCCCC(=O)NC1CCOC12CCCC2 |
N#CCCCNc1nc2c(c(NCCc3ccnc(O)c3)n1)CCC2 |
N#CCCN(CCN1CCOCC1)Cc1cccc(F)c1C(F)(F)F |
N#CCCSCC(=O)N(C[C@H]1C[C@@H]1c1cccs1)CC1(C2CC2)CC1 |
N#CCCSCC(=O)N1CSC[C@H]1C(=O)NCc1ccnc(CO)c1 |
N#CCc1ccc(CNS(=O)(=O)c2cc([N+](=O)[O-])ccc2C#N)cc1 |
N#CCc1ccsc1C(=O)N1CCCN(C(=O)[C@@H]2CNC(=O)O2)CC1 |
N#C[C@H]1CC[C@@H]1C(=O)NCC1(F)CN(c2nc3nc(Cl)ccc3s2)C1 |
N#C[C@H]1C[C@@H]1C(=O)NC(CC(=O)NCC1(n2nccn2)CC1)C(F)F |
N#C[C@H]1C[C@@H]1C(=O)NCc1ccc(C(=O)N[C@]23CC[C@H](C[C@@H]2O)C3)s1 |
N#C[C@H]1C[C@@H]1C(=O)NCc1ncccc1C(=O)NC1CCS(=O)(=O)C1 |
N#Cc1c[nH]c(C(=O)N2CC(C3(NC(=O)c4ccc(Cl)s4)CC3)C2)c1 |
N#Cc1c[nH]c(C(=O)N[C@H]2CC=CC[C@H]2C(=O)N[C@@H]2COC[C@H]2O)c1 |
N#Cc1cc(C(=O)N(CC(=O)N2CCCC3(CC3)C2)CC2CC2)cs1 |
N#Cc1cc(C(=O)NC[C@@H]2CCCN2C(=O)C2=C(Cl)CCOC2)c[nH]1 |
N#Cc1cc(C(=O)NCc2ccnc3[nH]ccc23)cc(C(F)(F)F)c1 |
N#Cc1cc(C(=O)N[C@H]2CC[C@H](C(=O)NCc3ccns3)CC2)c[nH]1 |
N#Cc1cc(CN(CC2C3CCCC32)C(=O)Cn2cc(Cl)cn2)cs1 |
N#Cc1cc(NCc2ccc3cc(F)c(F)cc3n2)ccc1C1CC1 |
N#Cc1cc2c([nH]1)CN(C(=O)Nc1ccc3c(Br)cccc3c1)CC2 |
N#Cc1ccc(C(=O)NCC2CCCCN2C(=O)C2CC=CC2)nc1 |
N#Cc1ccc(C(=O)NNC(=O)Cn2ccc(C(F)(F)F)n2)cc1Cl |
N#Cc1ccc(C=CC(=O)NCc2cccc(-n3cncn3)c2)cc1 |
N#Cc1ccc(CCC(=O)NC2CCc3cc(CN)ccc32)c(F)c1 |
N#Cc1ccc(CNC(=O)C2(F)CN(C(=O)CC3CC(F)(F)C3)C2)s1 |
N#Cc1ccc(CNC(=O)N2CCC3(CC2)OC[C@H](O)[C@@H]3O)c(F)c1 |
N#Cc1ccc(CNC(=O)Nc2cc(F)cc3c2CNC3=O)c(Br)c1 |
N#Cc1ccc(CNC(=O)[C@H]2CCN(C(=O)C(O)C3CC3)C[C@H]2O)s1 |
N#Cc1ccc(F)c(NNC(=O)N[C@H]2C[C@H]2Cc2ccc(Cl)cc2)c1 |
N#Cc1ccc(NC(=O)CCCOC(=O)CCCOC(F)(F)F)cc1 |
N#Cc1ccc(NC2CC2)c(NC(=O)c2cc(F)cc3cc[nH]c23)c1 |
N#Cc1ccc(NC2COCCCN(C(=O)Cc3ccns3)C2)nn1 |
N#Cc1ccc(NCC23COC(c4ccccc4)(C2)C3)cc1[N+](=O)[O-] |
N#Cc1ccc(S(=O)(=O)N2CCN(C(=O)Cc3cnoc3)CC2)cc1 |
N#Cc1ccc2c(c1)CCN(C(C(=O)NCC1CC1)c1cnc[nH]1)C2 |
N#Cc1ccc2ncc(C(=O)N3CCOc4cccc(Br)c4C3)n2c1 |
N#Cc1cccc(C(=O)N2C[C@H]3C[C@@]3(NC(=O)[C@]34CCC[C@H]3C4)C2)c1 |
N#Cc1cccc(C(F)(F)C(=O)NCCSCc2ccccc2F)c1 |
N#Cc1cccc(OC2CN(C(=O)c3cccc(C(N)CO)c3)C2)c1 |
N#Cc1ccccc1N1CCCN(C(=O)NCCC2CCOC2)CC1 |
N#Cc1ccccc1O[C@H]1CC[C@@H](NC(CF)c2ccccc2)CC1 |
N#Cc1csc(C(=O)N2CCCC2CNC(=O)CCCNC(N)=O)c1 |
N#Cc1oc2ccccc2c1NC(=O)CN1CCCC1c1cnco1 |
N#Cc1sccc1COC(=O)c1cnn(-c2cc(F)ccc2Cl)c1N |
NC(=O)C(=O)N1CCC2(CC(C(=O)NCCC3=CCCCCC3)C2)C1 |
NC(=O)C(=O)N1[C@@H]2CC[C@H]1C[C@H](NC(=O)CCc1cccc(=O)[nH]1)C2 |
NC(=O)C(F)(F)C1(O)CCN(C(=O)c2occc2-c2ccccc2)C1 |
NC(=O)C1(CNC(=O)NC2CCCN(c3cnccn3)C2)CCCC1 |
NC(=O)C1(NC(=O)C2(CCNC(=O)c3ccc(CO)cc3)CC2)CC1 |
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