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CNc1c(-c2sccc2I)nc2ccc3cc(C(=O)OC)ccc3n12
CNc1cc(-c2ccc(N3CCN(C)CC3)cc2)cc(C(F)(F)F)c1
CNc1cc(C(=O)N2CCOCC(NC(=O)CC=C(Cl)Cl)C2)ccn1
CNc1cc(C(=O)NC(C(=O)NCC2(CF)CC2)C2(C)CC2)ccn1
CNc1cc(N2CCC(CNC(=O)c3cnn(C)c3)CC2)nc(C)n1
CNc1ccc(-c2ccc3c(OC(F)F)nccc3c2)cc1[N+](=O)[O-]
CNc1ccc(C(=O)N(C)C2CC(C(=O)N3CC(C)(O)CO3)C2)nc1
CNc1ccc(C(=O)N2CSC[C@H]2C(=O)N2Cc3ncsc3C2)nc1
CNc1ccc(C(=O)N[C@@H](COC)C(=O)N[C@H]2C[C@H](O)C[C@@H]2O)nc1
CNc1ccc(F)cc1C(=O)NCc1ccc(-n2cc(Cl)cn2)cc1
CNc1ccccc1CNc1cc(N2CCC(C)S(=O)CC2)ncn1
CNc1ccnc(CNC(=O)NNC(=O)c2cc(F)c(F)cc2Cl)c1
CNc1cnccc1C(=O)NC(C(=O)NCC(=O)N(C)O)C1(C)CC1
CNc1nc(C(=O)N2CCN3CCOCC3(CO)C2)ccc1[N+](=O)[O-]
CNc1nc(N(C)CCC#N)nc(N2C[C@H]3CN(C(C)=O)C[C@H]3C2)n1
CNc1nc(NC(C)CC2CCOC2)nc(NC2CC3(CCC3)C2)n1
CNc1nc(NCc2cnn(C)c2)nc(NC2CCNC(=O)CC2)n1
CNc1nc(NCc2csc(Cl)c2)nc(NCc2cc(C)[nH]c2C)n1
CNc1ncc(C(=O)N(CC2CCSC2)CC2(C(C)(C)O)CCC2)o1
CNc1ncc(C(=O)N2CC[C@H]3[C@@H](C2)[C@@H]3NC(=O)CC2CC2(C)C)o1
CNc1ncc(C(=O)NC[C@H]2CCC[C@H]2NC(=O)[C@@H]2CCC[C@H]2O)o1
CNc1ncccc1C(=O)N1C[C@H]2C[C@@]2(C(=O)NCC2(CO)CC2)C1
CNc1ncccc1CNc1nccc(N(C)Cc2ccccn2)n1
CNc1scnc1C(=O)N1CC(=O)NCC1C(=O)N1CCC12CCC2
CNc1scnc1C(=O)N[C@H]1CCC[C@H](C(=O)NCC2=NOCC2)C1
COC(=O)/C=C/C1CCC(Nc2cccc(Cn3ccnc3C)c2)C1
COC(=O)C(C)(C)NC(=O)N1CC[C@H](OC)C[C@@H]1c1ccc(F)cc1
COC(=O)C(C)(C)NC(=O)NC1CC(=O)N(c2ccc(F)c(F)c2)C1
COC(=O)C(C)(C)ONC(=O)C(C)CNC(=O)CNC(=O)CN(C)C
COC(=O)C(C)(C)ONC(=O)CC[C@@H](C)NC(=O)c1nn(C)cc1Cl
COC(=O)C(C)(C)[C@@H](NC(=O)c1ccc2cc(I)ccc2n1)C(C)C
COC(=O)C(C)(C)c1cn(C2CN(C(=O)C3CC(=O)N(O)C3)C2)nn1
COC(=O)C(C)(CCF)NC(=O)C1CCn2cc(C(F)(F)F)nc2C1
COC(=O)C(C)(F)C(=O)NCC1CCN(C(=O)[C@H]2COCCO2)CC1
COC(=O)C(C)(F)C(=O)N[C@@H]1COC[C@H]1NC(=O)c1cncnc1C
COC(=O)C(C)(NC(=O)C[C@H](C)c1ccc2c(c1)OCO2)C1CCC1
COC(=O)C(C)(NC(=O)c1cncc(CCN)c1)c1ccc(F)cc1
COC(=O)C(C)C(=O)N1CC(SC)(C(=O)N(C)Cc2n[nH]c(C)n2)C1
COC(=O)C(C)C(=O)N1C[C@H](C)CC[C@H]1C(=O)N1CCOCC1CO
COC(=O)C(C)CC(=O)N(C)CCC(C)Nc1nc(C(F)(F)F)cs1
COC(=O)C(C)CC(=O)N[C@H]1CCC[C@@H](C(=O)N(C)c2ccsc2)C1
COC(=O)C(C)CN(C)C(=O)CCN(CCO)C(=O)C(C)C1CCC1
COC(=O)C(C)CNC(=O)CC(NC(=O)C(O)C1CCC1)C(C)(C)C
COC(=O)C(C)CNC(=O)c1oc(CNC(=O)c2cc[nH]n2)cc1C
COC(=O)C(C)COC(=O)c1ccc(COc2ccc(C#N)cc2)o1
COC(=O)C(C)N(C(=O)[C@H]1C[C@H]1CNC(=O)[C@H]1C[C@](C)(F)C1)C1CC1
COC(=O)C(C)N(C)C(=O)C1(N(C)C(=O)C2=CCC(C)(C)CC2)CC1
COC(=O)C(C)N(OC)C(=O)CCCCCNC(=O)c1cccnc1
COC(=O)C(C)NC(=O)C(CNC(=O)C(C)(C)n1cncn1)N(C)C
COC(=O)C(C)NC(=O)C1CC(C)(C)CCN1C(=O)C(F)C(C)(F)F
COC(=O)C(C)NC(=O)CCN(C(=O)CC1CCCN(C)C1)C1CC1
COC(=O)C(C)Nc1c(-c2ncoc2C)nc2cccc(C(N)=O)n12
COC(=O)C(C)ONC(=O)C1=C(F)CN(C(=O)CC(=O)N(C)C)CC1
COC(=O)C(C)ONC(=O)C1COCCN1C(=O)C1=C(C)OCCC1
COC(=O)C(C)ONC(=O)[C@H](CNC(=O)C(C)CCC(C)(C)C)OC
COC(=O)C(C)c1cccc(NC(=O)CC2CCN(C(C)C)CC2)c1
COC(=O)C(C)n1cc(C2CN(C(=O)c3ccn(C4CC4)n3)C2)nn1
COC(=O)C(CCF)NC(=O)C1=CCN(C(=O)c2[nH]cc(C)c2C)C1
COC(=O)C(CCc1cn[nH]c1)NC(=O)Cc1ccc2ocnc2c1
COC(=O)C(CNC(=O)Cc1nnc(OC)s1)Cc1ccc(Cl)cc1
COC(=O)C(CNC(=O)Nc1cc(SC)ncn1)c1ccc(F)cc1
COC(=O)C(Cc1ccccc1)N(C)C(=O)NC[C@@H]1[C@H](CO)C1(F)F
COC(=O)C(F)(F)CC1CN(C(=O)CCN(C)C2CCCCCC2)C1
COC(=O)C(F)(F)CNC(=O)[C@H]1CCC[C@H]1NC(=O)C1CCOCC1
COC(=O)C(F)Cc1ccc(NC(=O)N[C@@H](C)c2cnccn2)cc1
COC(=O)C(NC(=O)C1CCN1C(=O)[C@@H]([C@@H](C)O)N(C)C)C1CCC1
COC(=O)C(NC(=O)Cc1cc(C)c(Br)cc1C)c1ccc(C)nc1
COC(=O)C(NC(=O)N1CCCC(C(F)(F)F)CC1)c1ccccc1
COC(=O)C(NC(=O)c1ccc2cccc(F)c2n1)C1CS(=O)(=O)C1
COC(=O)C(NC(=O)c1cccc2cc[nH]c12)C1CCC(C)(C)CC1
COC(=O)C(NC(=O)c1nc(C(C)(F)F)cs1)c1cccc(F)c1O
COC(=O)C(NCC(C)(C)c1ccncc1F)c1ccc(F)cc1Cl
COC(=O)C(OC(=O)[C@H]1[C@@H]2CCCCC[C@@H]21)c1ccc(F)c(Cl)c1F
COC(=O)C(OC)C(=O)NCc1cc(C(=O)NC2CCCCC2)[nH]n1
COC(=O)C(c1cc(Cl)cc(Cl)c1)N1CC2(CCC2)OC2(CCC2)C1
COC(=O)C(c1ccc(C)cc1)N(C)C(=O)Nc1cccc(SC)c1
COC(=O)C1(C(=O)NC[C@H]2C[C@H]2NC(=O)[C@@H]2CCC[C@H](O)C2)CC1C
COC(=O)C1(C(=O)OC)CCN(CC(C)CCc2ccccc2)CC1
COC(=O)C1(C(NCCC(C)C)c2nnnn2CCC2(C)CC2)CC1
COC(=O)C1(C)CC(C(=O)N(C)C[C@H]2CCC[C@H]2Nc2ncns2)C1
COC(=O)C1(C)CC(NC(=O)C(CC2CCC2)NC(=O)[C@H]2C[C@@H]2C)C1
COC(=O)C1(C)CCCN(C(=O)CNS(=O)(=O)c2cn(C)c(C)n2)C1
COC(=O)C1(C)CCN1C(=O)[C@@H]1C=C[C@H](NC(=O)CC(C)C(F)F)C1
COC(=O)C1(C)CN(C(=O)c2nc(CNC(=O)C3CCO3)oc2C)C1
COC(=O)C1(CO)CN(Cc2ccc(Oc3ccc(Br)cn3)cc2)C1
COC(=O)C1(F)CCN(CCc2cn(-c3cccc(SC)c3)nn2)C1
COC(=O)C1(F)CCN(Cc2ccc(-c3ccccc3)cc2Cl)CC1
COC(=O)C1(N(C)C(=O)C(NC(=O)C2=CCCC2)c2ccoc2)CC1
COC(=O)C1(NC(=O)C2CN(C(=O)C(C)C#N)CC23CC3)CC(C)C1
COC(=O)C1(NC(=O)N2CC3(CC(c4ccccc4)C3)C2)CCCC1
COC(=O)C1(O)CN(C(=O)C2=CCC(NC(=O)c3cnccn3)C2)C1
COC(=O)C1(SC)CC(NC(=O)N2CCC[C@@]3(CO)CCCC[C@H]23)C1
COC(=O)C12CCC(C(=O)N3CCCC(C4CCNCC4)C3)(CO1)C2
COC(=O)C12CCC(CNC(=O)c3cn4c(n3)CC(C)CC4)(CC1)C2
COC(=O)C1=CCC(NC(=O)N2Cc3c(Br)cccc3C(C)(C)C2)C1
COC(=O)C1=NOC2(C1)CN(S(=O)(=O)c1cc3cncc(Br)c3o1)C2
COC(=O)C1C(C)CCN1C(=O)[C@H]1[C@@H]2CN(C(=O)c3ccc[nH]3)C[C@@H]21
COC(=O)C1C2CCCCC2C1NC(=O)N[C@H]1CCN(C2CCC2)C1
COC(=O)C1CC(=O)N(C2CN(C(=O)NC3CC34CC(C)(C)C4)C2)C1
COC(=O)C1CC(C)(C)CN1C(=O)c1ccnc(NC(=O)C(C)C)c1