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COc1c(C(=O)N2Cc3ccccc3CCC23CCC3)occc1=O
COc1c(C(=O)NCC(O)CNS(=O)(=O)C2CC=CC2)ccnc1F
COc1c(C(=O)NCc2cnn(C)c2C(F)(F)F)ccc2c1CCC2
COc1c(C)cccc1CNC(=O)Nc1nnc(C2CCCCO2)s1
COc1c(Cl)cc(C(=O)OC[C@@H](O)COCc2ccccc2)cc1Cl
COc1c(Cl)cc([N+](=O)[O-])cc1CNC(c1cccc(C)n1)C1CC1
COc1c(Cl)ccc(Cl)c1COC(=O)C1CSCN1C(=O)C1CCC1
COc1c(Cl)ccc2c1CN(C(=O)NC(C(C)(C)C)C(C)(C)C)CC2
COc1c(Cl)ccnc1CN(CCC1(O)CCC1)CC1CCC(C)C1
COc1c(F)c(F)cc(CNC(=O)C(CCC(C)C)NC(C)=O)c1F
COc1c(F)cc(CNC(=O)N[C@@H](CO)c2cccc(Cl)c2)cc1F
COc1c(F)cc(S(=O)(=O)N[C@H](C)C(=O)Nc2ccccc2)cc1F
COc1c(F)ccc(F)c1C(=O)N1CCC(NC(=O)C(F)(F)F)CC1
COc1c(F)ccc(F)c1CNC(=O)N(C)C1(c2cccnc2)CC1
COc1c(F)ccc2[nH]c(C(=O)N3CCCN(CCC#N)CC3)cc12
COc1c(F)cccc1CN(CC1CC2(CC2)C1)C(=O)C(C)CSC
COc1c(NC(=O)N2CCc3ccc(Cl)c(F)c3C2)ccc(F)c1F
COc1c(NC(=O)[C@@H]2CC[C@@H]2NC(=O)[C@H](C)NC(C)=O)c(C)nn1C
COc1cc(-c2cccc(C(=O)CC(F)(F)F)c2)cc2c1OCCO2
COc1cc(-c2noc(-c3cc4oc(C)cc4[nH]3)n2)cc(Cl)c1OC
COc1cc(-n2cnnn2)c(Cl)cc1C(=O)OCCc1cc(C)on1
COc1cc(Br)c(C(=O)N[C@H](C)c2ccc3c(c2)CCC3)cc1OC
COc1cc(Br)cc(C(=O)N(Cc2ccccc2)OCC(C)C)c1O
COc1cc(Br)cc(OC)c1CC(=O)NC1CCN(CCCO)CC1
COc1cc(C#N)ccc1CNC(=O)NCc1c(C)nn(C)c1OC
COc1cc(C#N)ccc1NC(=O)NCC(OC)c1ccccc1C
COc1cc(C(=O)N(C)C[C@H](C)NC(=O)c2cc(F)ccc2N)n[nH]1
COc1cc(C(=O)N(CCNC(=O)C2(F)CC=CC2)C2CC2)ccn1
COc1cc(C(=O)N(Cc2ccc(C)s2)CC23CCC(CC2)C3)sn1
COc1cc(C(=O)N2CC(C(O)C(=O)NCc3ocnc3C)C2)n[nH]1
COc1cc(C(=O)N2CC(OCc3nc(C)no3)C2)cc(OC)c1C
COc1cc(C(=O)N2CC=CC(C(=O)N(C)C34CC(C3)C4)C2)n(C)n1
COc1cc(C(=O)N2CC=CC2C(=O)N2CCC(C)C(F)(F)C2)on1
COc1cc(C(=O)N2CCCC(OC)(C(F)F)C2)nc2ccccc12
COc1cc(C(=O)NC(C(=O)N2CCC(C)(C#N)C2)C(C)(C)C)on1
COc1cc(C(=O)NC(C)Cc2cc(C)cc(C)c2)cc2cn[nH]c12
COc1cc(C(=O)NC2(C(=O)N3CC[C@@H]4[C@H]3C[C@H]4OC)CC2)ncn1
COc1cc(C(=O)NC2CC(NC(=O)C(C)N3CCOC3=O)C2)sn1
COc1cc(C(=O)NCC2=CCCN(C(=O)C(F)=CC3CC3)C2)sn1
COc1cc(C(=O)NCC2CC(CNC(=O)c3cnsn3)C2)ccn1
COc1cc(C(=O)NCCC(OC)C(C)C)ccc1OC1CCCC1
COc1cc(C(=O)NCCCC(C)NC(=O)Cc2ccno2)nn1C
COc1cc(C(=O)NC[C@H](CO)NC(=O)C2(C)CCC3CC3C2)on1
COc1cc(C(=O)NCc2occc2C(=O)NCC(C)(C)SC)n[nH]1
COc1cc(C(=O)N[C@@H](C)c2nc(-c3cccnc3)cs2)cnc1Cl
COc1cc(C(=O)N[C@H]2CN(C(=O)c3c(C)csc3C)C[C@H]2F)on1
COc1cc(C(=O)Nc2c(C#N)oc3ccccc23)ccc1[N+](=O)[O-]
COc1cc(C(=O)Nc2cnc3c(c2)CC(C)CC3)ccc1C(=O)O
COc1cc(C(=O)O)nc(C(=O)N2CCc3ccc(F)cc3C2C)c1
COc1cc(C(=O)OCCOCCC(=O)OC(C)(C)C)c(F)cc1Br
COc1cc(C(=O)OCc2cncc(C(C)(F)F)c2)ccc1C(F)F
COc1cc(C(C(=O)NC2CC2)N2CCOCC2(C)C)c(F)cc1F
COc1cc(C(F)(F)F)ccc1C(=O)NCC(CC(C)(C)C)C(=O)O
COc1cc(C(F)(F)F)ccc1CNC(=O)NNC(=O)NCC(F)F
COc1cc(C(F)F)ccc1CN1CCC(CCNS(N)(=O)=O)CC1
COc1cc(C)c(Br)c(C)c1S(=O)(=O)NC[C@H](O)CN1CCCCC1
COc1cc(C)c(CN(C)C(=O)NCCc2cc(C)on2)cc1OC
COc1cc(C)c(CN2CC3(CCN(C)CC3)c3ccccc32)cn1
COc1cc(C)c2c(c1)NC(C(=O)N1CC(S(C)(=O)=O)CCC1C)C2
COc1cc(C)c2cc(C(=O)Nc3ccc(C)c(C4CC4)c3)[nH]c2c1
COc1cc(C)cc(C)c1C(=O)COC(=O)CN1CC(C)CS1(=O)=O
COc1cc(C)cc(CC(=O)NC[C@H](CF)NS(=O)(=O)CC2CC2)c1
COc1cc(C)cc(CN(CC2(Cl)CC2(F)F)C(=O)[C@H]2CC2(F)F)c1
COc1cc(C)cc(CN(CCOCCSC)C(=O)C2CCCC2)c1
COc1cc(C)ccc1C(=O)NCCN(C(=O)CC1CSC1)C1CC1
COc1cc(C)ccc1NC(=O)[C@@H]1[C@H](C)CN1C(=O)C(F)C(F)(F)F
COc1cc(C)ccc1NC(=O)[C@]12CCC[C@H]1CN(C(=O)CC#N)C2
COc1cc(C)ccc1OCC(=O)NCc1ccc2ccn(C)c2c1
COc1cc(C)cnc1CN[C@H](CO)CCCNC(=O)OC(C)(C)C
COc1cc(C)ncc1C(N[C@H]1CC[C@H](CO)CC1)c1nnnn1C
COc1cc(C2CC2)ccc1NC(=O)N1CCC(C)(CS(C)(=O)=O)C1
COc1cc(C2CCN(C(=O)C(O)C(C)(C)C)C2)ccc1C(F)(F)F
COc1cc(C2CCN(C(=O)NC3COC(C)(C)C3)C2)cc(F)c1F
COc1cc(C=CC(=O)NCC(=O)NC2CNC2)cc(OC)c1OC
COc1cc(C=Cc2nc(-c3ccccc3)cs2)ccc1OCC#N
COc1cc(CC(=O)NNc2nc(C)ccc2[N+](=O)[O-])cnc1OC
COc1cc(CC(=O)Nc2ccc(N3CCCC(C)C3)c(Cl)c2)on1
COc1cc(CC(C)NC(=O)c2cc3ccc(C)cn3n2)ccc1O
COc1cc(CCC(=O)NCCC(C)NS(=O)(=O)C2(C)CC2)ccn1
COc1cc(CCC(=O)NCCCc2cccc(C)c2)cc(OC)c1
COc1cc(CCNC(=O)N(C)C2(c3cccnc3)CC2)cc(C)n1
COc1cc(CN(C)C(=O)c2cc3cccnc3nc2C)ccc1C
COc1cc(CN(C)C)ccc1NC(=O)c1cnc2ccc(F)cn12
COc1cc(CN(C=O)[C@H](C)c2ccc3c(c2)CCCC3)c(F)cn1
COc1cc(CN(CC(C)(C)OC)C(=O)CCCC(C)=O)c(F)cn1
COc1cc(CN(CC(C)OC(F)F)C(=O)[C@H]2CNC(=O)C2)ccn1
COc1cc(CN(CC(CO)C2CC2)C(=O)C(C)(O)C(F)(F)F)sn1
COc1cc(CN(Cc2cc(Br)[nH]n2)Cc2ccc(Cl)o2)c(Cl)cn1
COc1cc(CN(Cc2cc(C)c(C)cc2C)CC(F)C2CC2)sn1
COc1cc(CNC(=O)C2C=CCN(C(=O)C3=COCCC3)C2)on1
COc1cc(CNC(=O)C2CCCCN2C(=O)C2=CCN(C)C2)on1
COc1cc(CNC(=O)Nc2ccc3ncsc3c2)cc(O)c1OC
COc1cc(CNC(=O)[C@H](C)n2cc(C3CCC3)nn2)c(Br)cc1C
COc1cc(CNC(=O)c2c(F)cc(F)c(O)c2F)cc(O)c1OC
COc1cc(CNC(=O)c2cnn3c2SCC3)ccc1OCC(N)=O
COc1cc(CNC2CCN(Cc3cccc(F)c3)CC2)ccc1F
COc1cc(CNCC2CC2(Br)Br)ccc1OCCN1CCOCC1
COc1cc(CNCc2ccc(C(F)(F)F)cc2C)cc(C(=O)O)c1
COc1cc(CNCc2cccc(S(C)(=O)=O)c2)ccc1OC(F)F
COc1cc(CNc2ccc(OCCN(C)C)cc2OC)ncc1Cl