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COc1cccc(C(O)CN2CCC(c3cc(C)cc(C)c3)CC2)c1
COc1cccc(C)c1CN(CC[C@H]1CC[C@H]1C)C(=O)c1ccns1
COc1cccc(C)c1CNC(=O)N(C)Cc1c(C)nn(C)c1OC
COc1cccc(C2(C)CCN(Cc3cc(F)c(OC)cc3F)C2)c1
COc1cccc(C2(CNC(=O)COc3c(F)cccc3F)CC2)n1
COc1cccc(C2(CNC(=O)Nc3cnccc3C#N)CCC2)n1
COc1cccc(CC(=O)N2C[C@H](NC(=O)C3CSC3)[C@H](OC)C2)c1
COc1cccc(CN(CC(C)C2CC2)C(=O)c2ncccc2Cl)n1
COc1cccc(CN(Cc2cc(Cl)cc(C#N)c2)C[C@H]2C[C@H]2C)n1
COc1cccc(CNC(=O)c2ccc(C#N)cc2O)c1OC(F)F
COc1cccc(F)c1C(=O)NC1CC(NC(=O)c2coc(C)c2)C1
COc1cccc(NC(=O)CN(c2ccc(OC)c(F)c2)C(C)C)c1
COc1cccc(NC(=O)NCCCn2cc(P(C)(C)=O)cn2)c1F
COc1cccc(NC(=O)[C@@H](NC(=O)[C@@H]2CC[C@H]2C#N)C(C)C)c1F
COc1cccc(OC(F)(F)F)c1C(=O)NCCC1(C(F)(F)F)CC1
COc1cccc(OC)c1CC(=O)NC1(c2nn[nH]n2)CCSCC1
COc1cccc(S(=O)(=O)NC[C@H]2CC[C@H]2NC(=O)c2ccon2)c1
COc1cccc2c(=O)[nH]c(N3CCCCNC(=O)C(F)(F)C3)nc12
COc1cccc2c(C)c(C(=O)N3CCn4c(C)nnc4C3C)oc12
COc1cccc2c1CC(c1nc(-c3cnn(CCO)c3)no1)CO2
COc1cccc2c1CCCC2(O)CNC1CC2(C1)CC(C)(C#N)C2
COc1cccc2c1CCCN(C(=O)C[C@H]1C[C@]3(CCNC3)CO1)C2
COc1cccc2c1N(CC(=O)COc1ccc(F)cc1)CCN2C
COc1cccc2c1OCC(C(=O)N1CC(C)(N3CCNCC3)C1)C2
COc1cccc2cc(-n3cc(-c4c(C)nn(C)c4Cl)nn3)cnc12
COc1ccccc1-c1cccc(NC(=O)C(C)c2ccnn2C)c1
COc1ccccc1-n1nccc1CN(C=O)CCC1CC=CCC1
COc1ccccc1C(=O)N(C)CCNC(=O)N1C[C@H]2COC[C@H]2O1
COc1ccccc1C(=O)N1CC=C(C(=O)N[C@H](CCO)C(C)C)C1
COc1ccccc1C(=O)N[C@@H](C)CCC(=O)N[C@@H](C)CS(C)(=O)=O
COc1ccccc1C(C)(C)C(=O)NCCc1c(Br)cccc1OC
COc1ccccc1C(C)N(C)C(=O)c1ccc2c(c1C)NCCO2
COc1ccccc1C(C)NC(=O)NCc1c(C)c(C)cc(C)c1C
COc1ccccc1C(O)CNC(=O)NCCc1cccc(C)c1Cl
COc1ccccc1C1(C(=O)N2CCCC(F)(C(N)=O)C2)CCCC1
COc1ccccc1C1(CNC(=O)[C@@H]2CSCC(=O)N2)CCOCC1
COc1ccccc1CC(C)CC(=O)N1CC(N2CCCOCC2)C1
COc1ccccc1CC(C)CC(=O)NC1CCc2cccc(O)c21
COc1ccccc1CCCNCCCc1cccc(C(F)(F)F)c1
COc1ccccc1CN(C)C(=O)c1ccccc1OC1CCCC1
COc1ccccc1CN1CCN(C(=O)c2cn3c(n2)CCC3)CC1
COc1ccccc1CNC(=O)C(C)N1CCC(CCCCO)CC1
COc1ccccc1COCC(O)COC(=O)CCn1ccnc1C
COc1ccccc1C[C@@H](C)NC(=O)Cc1cccc2c1CCCC2
COc1ccccc1N(C)C(=O)C1CCCN1C(=O)C(SC)C(C)C
COc1ccccc1N(CCC#N)C(=O)C(C)NC1(C)CC(OC)C1
COc1ccccc1OCC(O)CNCC1(C(=O)OC(C)(C)C)CC1
COc1ccccc1[C@H]1C[C@H](NC(=O)N2CCC3(CC(OC)C3)C2)C1
COc1cccnc1CNC(=O)CC(NC(=O)CCSC)C(C)(C)C
COc1ccn2c(CNC3CCS(=O)(=O)c4ccccc43)cnc2c1
COc1ccnc(C(=O)Nc2cccc(C#Cc3cccs3)c2)c1O
COc1ccnc(CNC(=O)C2(C)CCN(C(=O)CC3CC3)CC2)c1
COc1ccnc(CNC(=O)[C@@H]2C[C@@H](C)CN2C(=O)c2ccco2)c1
COc1ccnc(N2CCC(C(=O)Oc3cc(Br)ccc3F)CC2)n1
COc1ccnc(N2CCN(C(=O)Nc3cnc(Cl)c(C)c3)CC2)c1
COc1ccnc(N2CCN(c3ncc(C#N)cc3[N+](=O)[O-])CC2)n1
COc1ccncc1C(=O)N1CC(C)(C(=O)NCc2coc(C)c2)C1
COc1ccncc1C(=O)N1CC[C@H](F)C[C@@H]1C(=O)NCCC1CC1
COc1ccsc1C(=O)NC[C@H]1CC[C@@H](C(=O)N2C3CSCC2C3)O1
COc1ccsc1C(=O)N[C@H]1C[C@@H](NC(=O)CCCCNC(C)=O)C1
COc1ccsc1CN(CC1C(F)(F)C12CCC2)C(=O)c1cocn1
COc1cnc(CN(CC2(C(C)C)CCCC2)C(=O)C2CSC2)nc1
COc1cnc(CNC(=O)[C@@H](NC(=O)C2CC3CC3C2)C(C)C)cn1
COc1cnc(CNC(=O)c2cccc(-c3ccccn3)c2C)cn1
COc1cnc(F)c(NC(=O)Nc2ccc3nc(S(C)=O)[nH]c3c2)c1
COc1cnc(N[C@H](CO)CNC(=O)CCCC(C)(C)C)nc1CO
COc1cncc(-c2cn([C@@H](C)CNC(=O)C3(C)CCCC3)nn2)n1
COc1cncc(C(=O)N(CCC(=O)NCC2CC(C)C2)C2CC2)n1
COc1cncc(C(=O)N(CCCNC(=O)c2cc[nH]n2)C2CC2)n1
COc1cncc(C(=O)N2C[C@H](O)C[C@H]2C(=O)N2CCC(C)CC2)n1
COc1cncc(C(=O)NC2CCN(C(=O)C#CC3CC3)CC2F)n1
COc1cncc(C(=O)NCCc2nc(-c3cnccn3)no2)c1C
COc1cncnc1C(=O)NC[C@@H](C)Nc1cc(S(C)(=O)=O)ncn1
COc1cncnc1NC(=O)c1ccc(-c2cccc(C#N)c2)cc1
COc1cnnc(C(=O)NC2(C(=O)NCc3cnns3)CC(O)C2)c1
COc1cnnc(C(=O)NC2CCN(C(=O)C3=C(C)CCC3)CC2)c1
COc1cnnc(C(=O)NCc2ccc(C(=O)N3CC(O)C3)cc2)c1
COc1cnncc1C(=O)N1CC(CNC(=O)C2(C)CCCC2C)C1
COc1csc(C(=O)N[C@H]2C[C@H]2CNC(=O)c2cc(=O)n(C)cn2)c1
COc1cscc1C(=O)NC(C(=O)NC[C@H](CO)OC)c1cccs1
COc1cscc1C(=O)N[C@@H](CCC(=O)NCC(C)(C)OC)C(C)C
COc1n[nH]cc1C(=O)NC(C(=O)N1CCC12CCC2)c1cccs1
COc1n[nH]cc1C(=O)NCC1(CC(=O)N2CCC3(CCO3)C2)CC1
COc1n[nH]cc1CN(CC1(C(C)C)CC1)C(=O)C1(CCF)CCC1
COc1n[nH]cc1CN(CCCc1ccco1)CC(OC)C(F)(F)F
COc1nc(C(=O)NC[C@H]2CCCN(C(=O)[C@H]3CC3(C)C)C2)sc1C
COc1nc(C)ccc1C(=O)NC1CCCN(c2cccc(C)c2)C1
COc1nc(C)ccc1CNC(=O)N[C@H]1C[C@@H]1c1cccc(F)c1F
COc1nc(C)ccc1CNS(=O)(=O)C1CC(C(=O)OC(C)(C)C)C1
COc1nc(C)sc1C(=O)NC/C=C\CNC(=O)C(C)OCC1CC1
COc1nc(C)sc1C(=O)NCCCCNS(=O)(=O)C1CCCC1C
COc1ncc(C(=O)N2CC(CNC(=O)c3nscc3C)(OC)C2)s1
COc1ncc(C(=O)N2CCCC2C(=O)NCCCC(=O)N(C)C)s1
COc1ncc(C(=O)NC(C)CCCNC(=O)c2cn[nH]c2C)cn1
COc1ncc(C(=O)NC(CN(C)C)C(=O)NCC(C)C2CC2)cn1
COc1ncc(C(=O)NC23CC(NC(=O)C4=NOC(C)(C)C4)(C2)C3)s1
COc1ncc(C(=O)NCC2(CNC(=O)c3ccoc3C)CC2)cn1
COc1ncc(F)c(N[C@@H](CF)CNC(=O)C2CCCC(C)N2C)n1
COc1ncc(F)cc1-c1cn(CCC(=O)NCCCC(F)F)nn1
COc1ncc(NC(=O)C(=O)NCCCS(=O)(=O)C(F)(F)F)cc1Br