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Cc1ncc(C(=O)N2CCN(C(=O)C3CC3(Cl)Cl)C[C@H]2CO)c(C)n1 |
Cc1ncc(C(=O)NC2(C(=O)N3CC(C)OCC(C)(C)C3)CSC2)o1 |
Cc1ncc(C(=O)NC2CC=C(C(=O)NCC[C@@H]3CCC[C@H]3O)C2)s1 |
Cc1ncc(C(=O)N[C@H](C(=O)NOCC(C)(C)C)[C@@H](C)O)cc1C#N |
Cc1ncc(C(=O)N[C@H](C)C2CN(C(=O)c3cnn(C)c3C)C2)cn1 |
Cc1ncc(C(=O)N[C@H](Cc2csc(NCCCO)n2)CC(C)C)o1 |
Cc1ncc(C(=O)N[C@H]2COC[C@H]2NC(=O)c2oncc2C)c(C)n1 |
Cc1ncc(C(=O)N[C@H]2C[C@H](NC(=O)C(C)(C)CC(F)F)C2)c(N)n1 |
Cc1ncc(C(=O)OCc2ccc(Br)c3cccnc23)c(C2CC2)n1 |
Cc1ncc(CC(=O)N2CCC(C(=O)NC3CCCC3C#N)C2C)s1 |
Cc1ncc(CC(=O)NC2CC(CNC(=O)C(C)C(F)F)C2)c(O)n1 |
Cc1ncc(CCCNC(=O)NCCOc2ccccc2C(C)C)[nH]1 |
Cc1ncc(CCNC(=O)C2(NC(=O)CC3CCCO3)CC(O)C2)s1 |
Cc1ncc(CN(CCOCC(F)(F)F)C(=O)C2CCCN2C)n1C |
Cc1ncc(CN(CCc2cccnc2)C(=O)C2CCCC(F)C2)s1 |
Cc1ncc(CN(C[C@H]2COC(C)(C)O2)C(=O)[C@H]2CCC(=O)O2)n1C |
Cc1ncc(CN(Cc2ccc(C(C)(C)O)cc2)CC2(C)CC2C)s1 |
Cc1ncc(CN(Cc2cn(C)nn2)CC2(C)CC3(CC3)C2)cc1Cl |
Cc1ncc(CN(Cc2cncc(Cl)c2)CC2(CF)CCCOC2)s1 |
Cc1ncc(CNC(=O)[C@H]2C[C@@H]2C(C)NC(=O)CCC(=O)N(C)C)o1 |
Cc1ncc(CNC(CCc2ccccc2)c2ccc(C)c(F)c2)o1 |
Cc1ncc(N)cc1C(=O)N[C@@H](C)CCNC(=O)COC1CCCC1 |
Cc1ncc(NC(=O)CC2CCCN2C(=O)CCC2CC2)cc1C#N |
Cc1ncc(NC(=O)NCc2ccc3c(c2)C(=O)NCC3)cc1C#N |
Cc1ncc(NC(=O)[C@@H](O)CNC(=O)c2cc(Cl)cn2C)c(C)c1C |
Cc1ncc(NC(=O)[C@H]2CCC[C@H]2NC(=O)c2ccn(C)c2)cc1Cl |
Cc1ncc(S(=O)(=O)N2CC3(CC(CNC(=O)/C=C/C(F)F)C3)C2)s1 |
Cc1ncc(S(=O)(=O)NC2CCC(C)(CNC(=O)CCC3CC3)C2)[nH]1 |
Cc1ncc2c(n1)CN(C(=O)NCc1cn(C3CCOC3)nn1)CC2 |
Cc1nccc(C(=O)N2CCC=CC2C(=O)NCCCCCCF)n1 |
Cc1nccc(C(=O)N[C@H](C)C(=O)N(C)Cc2ccc(O)cc2)c1N |
Cc1nccc(CCNC(=O)[C@H]2CC[C@H](CNC(=O)C3CC3)CC2)n1 |
Cc1nccc(NC(=O)N2CC3(CCCCC3)c3ccccc32)c1C |
Cc1nccc(NCCNC(=O)N2CC(Cc3ccccc3O)C2)n1 |
Cc1ncccc1C(=O)N1CCC(C(=O)NCCOCC2CC2)CC1 |
Cc1ncccc1C(=O)N1CCC(OCCNC(=O)OC(C)(C)C)C1 |
Cc1ncccc1C(=O)NNC(=O)NCC1(C(F)(F)F)CC(F)(F)C1 |
Cc1ncccc1C(=O)N[C@H](C(=O)NC1CC(C(F)F)C1)C(C)(C)C |
Cc1ncccc1CC(=O)N(CC(=O)NC12CCCCC1C2)C1CC1 |
Cc1ncccc1CC(=O)N1CCC(C)(C)C1C(=O)N1CC2CC2C1 |
Cc1ncccc1CC(=O)N1CCC1C(=O)N1CC2CC3CC2C1C3 |
Cc1ncccc1CNC(=O)[C@@H](NC(=O)C12C=CC(CC1)C2)C(C)C |
Cc1nccn1-c1ccncc1NC(=O)c1cccc2ccncc12 |
Cc1nccn1C(C)C(=O)N1C[C@@H](F)C[C@@H]1C(=O)NC[C@@H]1CCCO1 |
Cc1nccn1CCCc1nc(-c2ccnc(-n3ccnc3)c2)no1 |
Cc1nccn1CCNC(=O)C1CCN(C(=O)c2ncccc2O)C1 |
Cc1nccn1CCNC(=O)[C@H](NC(=O)C(O)C(C)(C)C)C(C)(C)O |
Cc1nccnc1C(=O)N1C[C@H]2C[C@@H]1[C@H]2C(=O)NCCC1C=CCC1 |
Cc1nccnc1CCNC(=O)C(CC1CC1)NC(=O)[C@@H]1C[C@H]1C#N |
Cc1nccnc1CCNC(=O)C1CCN(C(=O)C2CSC2)C12CC2 |
Cc1nccnc1CNCCC(CC(C)(C)C)NC(=O)OC(C)(C)C |
Cc1nccnc1N1CCN(C(=O)C(=O)N2C[C@H](C)O[C@@H](C)C2)CC1 |
Cc1ncn(O)c1C(=O)NC1COCCN(C(=O)c2ccoc2C)C1 |
Cc1ncnc2c1CN(Cc1cc(-c3ccncc3)ccc1Cl)CC2 |
Cc1ncncc1C(=O)N1CC2(CC(NC(=O)[C@H]3CC[C@H]3C#N)C2)C1 |
Cc1ncncc1C(=O)NC(C)(C)CCC(=O)N(C)[C@H](C)CN(C)C |
Cc1ncncc1C(=O)NCC1CCCN(C(=O)c2cnccn2)C1 |
Cc1ncncc1NC(=O)c1ccc(CNC(=O)C(F)=CC2CC2)s1 |
Cc1ncoc1-c1ccc(NC(=O)C[C@@H](N)CC2CCCCC2)cc1 |
Cc1ncoc1C(=O)N(CCN(C)C(=O)CC1CCOCC1)C(C)C |
Cc1ncoc1C(=O)N1CCO[C@H](C(=O)NCCNC(=O)C2CC2)C1 |
Cc1ncoc1C(=O)N1C[C@@H](F)C[C@H]1C(=O)N(C)Cc1cnccn1 |
Cc1ncoc1C(=O)N[C@H]1CC[C@H](NC(=O)c2cc(CO)n(C)n2)C1 |
Cc1ncoc1CN(Cc1cc(C(C)(C)C)no1)Cc1[nH]ncc1Br |
Cc1ncoc1CNC(=O)NCC1(c2ccc(Br)cc2)CCOCC1 |
Cc1ncsc1C(=O)N1CCO[C@@H](C)[C@@H]1C(=O)NCc1ccncc1 |
Cc1ncsc1C(=O)NC[C@H](NC(=O)C(C)(C)C1CCOC1)C(C)C |
Cc1ncsc1C(=O)N[C@@H]1CCCN(C(=O)C2CCCC(F)(F)C2)C1 |
Cc1ncsc1C(=O)N[C@H]1CCCC[C@H]1CC(=O)N[C@@H]1COC[C@H]1F |
Cc1ncsc1C(C)NC(=O)C(C)(C)CCCNC(=O)[C@H]1C[C@H]1C#N |
Cc1ncsc1CC(=O)N[C@@H](CC(C)(C)C)C(=O)NCC(C)CCO |
Cc1ncsc1CC(=O)N[C@H]1CC[C@@H](CC(=O)N(C)CCCO)CC1 |
Cc1ncsc1CCCN(C)c1nccc(N2CCCC(C)(C)C2)n1 |
Cc1ncsc1CCN(Cc1ccc(F)cc1O)C(=O)C1(CF)CC1 |
Cc1ncsc1CCNc1nc(NCC2(F)CCC2)nc2cc[nH]c12 |
Cc1ncsc1CCOC(=O)CCc1nc(O)c2cc(F)ccc2n1 |
Cc1ncsc1CN(Cc1cn(C)cn1)C[C@]1(F)CC[C@@H](CO)CC1 |
Cc1ncsc1S(=O)(=O)NCCCCN(C)C(=O)c1cnc(S)nc1 |
Cc1nn(-c2ccccc2)c(NC(=O)N2C3CCC2(CO)CC3)c1C |
Cc1nn(C(C)(C)C)c(C)c1NC(=O)NCC1CCC2(C1)CC2(F)F |
Cc1nn(C(C)C)c(NCCc2c[nH]c3cccc(C)c23)c1[N+](=O)[O-] |
Cc1nn(C)c(Cl)c1CN(CC(C)(C)CO)C(=O)C1COCC(C)O1 |
Cc1nn(C)c(N)c1C(=O)NCC1CCN1C(=O)c1ncncc1Cl |
Cc1nn(C)c(N)c1C(=O)N[C@H]1C[C@H]1NC(=O)COc1cccnc1 |
Cc1nn(C)c(NC(=O)c2ccc3c(c2)N(C)CCC3)c1C(F)(F)F |
Cc1nn(C)c2c(N(C)CCCO)nc(N(C)CCOC3CC3)nc12 |
Cc1nn(C)c2c(N3CCN(c4ccc(F)cn4)CC3)nc(Cl)nc12 |
Cc1nn(C)c2c(NCCC3CC3)nc(NCCCCC(N)=O)nc12 |
Cc1nn(C)c2sc(C(=O)Nc3ncc(-c4ccc(F)cc4)s3)cc12 |
Cc1nn(C)cc1C(=O)NC(CC(=O)NCC(=O)NCCO)C(C)C |
Cc1nn(C)cc1C(=O)NCCC1CCN(Cc2ccccc2)CC1 |
Cc1nn(C)cc1C(=O)N[C@H]1C[C@@H]2C[C@H]1[C@H](NC(=O)C1CC(F)C1)C2 |
Cc1nn(C)cc1C(C)NC1C[C@@H]2CN(C(=O)OC(C)(C)C)C[C@@H]2C1 |
Cc1nn(C)nc1C(=O)N1CCCCC(CNC(=O)C2=CCSC2)C1 |
Cc1nn(C)nc1C(=O)NCC(C)(C)CN(C)C(=O)CC1C=CCC1 |
Cc1nn(C2CC2)cc1C(=O)NCC[C@@H](C)NC(=O)C1(O)CCOC1 |
Cc1nn(C2CCCCC2)cc1C(=O)N1CCC(C2(O)CCC2)CC1 |
Cc1nn(CC(=O)N2CCC(N3C(=O)CCC3=O)C2)c2ncccc12 |
Cc1nn(CC(=O)N2C[C@H](C)CC[C@@H]2C(=O)N2CCSCC2)c(=O)o1 |
Cc1nn(CC(=O)NCC[C@H]2C[C@H](NC(=O)C3CCCC3)C2)c(=O)o1 |
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