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COc1c(C#N)cccc1CC(=O)N(C)c1nnn(C)c1C(F)(F)F
COc1c(C#N)cccc1CNc1cc(-c2ccccc2C)nn1C
COc1c(C(=O)N2CCN(C(=O)c3ccco3)C(C)C2C)csc1C
COc1c(C(=O)N2Cc3ccccc3CCC23CCC3)occc1=O
COc1c(C(=O)NCc2cnn(C)c2C(F)(F)F)ccc2c1CCC2
COc1c(C(=O)Nc2ccc(C3CC3)c(-c3nn[nH]n3)c2)csc1C
COc1c(C)cc(Cl)cc1NC(=O)c1cc(-c2ccccc2)nn1C
COc1c(C)cc(Cl)cc1NCc1cccc(C(=O)NCC(C)C)c1
COc1c(C)cccc1CNC(=O)Nc1nnc(C2CCCCO2)s1
COc1c(Cl)ccc(Cl)c1COC(=O)C1CSCN1C(=O)C1CCC1
COc1c(Cl)ccc2c1CN(C(=O)NC(C(C)(C)C)C(C)(C)C)CC2
COc1c(Cl)ccnc1CN(CCC1(O)CCC1)CC1CCC(C)C1
COc1c(F)c(F)cc(CNC(=O)C(CCC(C)C)NC(C)=O)c1F
COc1c(F)c(F)cc(CNc2cc(N3CCNCC3)ccn2)c1F
COc1c(F)cc(S(=O)(=O)N[C@H](C)C(=O)Nc2ccccc2)cc1F
COc1c(F)ccc(F)c1CNC(=O)N(C)C1(c2cccnc2)CC1
COc1c(F)ccc2[nH]c(C(=O)N3CCCN(CCC#N)CC3)cc12
COc1c(F)cccc1CN(C)C(=O)NC(c1ncccn1)C1CC1
COc1c(F)cccc1CN(C)S(=O)(=O)CCOCc1ccccc1
COc1c(F)cccc1NC(=O)C/C=C/CNC(=O)CCP(C)(C)=O
COc1c(NC(=O)[C@@H]2CC[C@@H]2NC(=O)[C@H](C)NC(C)=O)c(C)nn1C
COc1cc(-c2ccc(O)c(NC(=O)OC(C)(C)C)c2)cn(C)c1=O
COc1cc(-c2nc(-c3ccc(CC(C)C)[nH]c3=O)no2)ccc1C
COc1cc(-n2cnnn2)c(Cl)cc1C(=O)OCCc1cc(C)on1
COc1cc(=O)n(C)cc1C(=O)NCc1nc2cc(C)ccc2n1C
COc1cc(Br)c(C(=O)N[C@H](C)c2ccc3c(c2)CCC3)cc1OC
COc1cc(Br)c(CN(C=O)CC2CCC3(CCC3)OC2)cc1OC
COc1cc(C#N)cc(CNc2ncc(S(=O)(=O)C(F)(F)F)cn2)c1
COc1cc(C#N)ccc1CCC(=O)OCCC=Cc1ccccc1
COc1cc(C#N)ccc1CNC(=O)NCc1c(C)nn(C)c1OC
COc1cc(C#N)ccc1NC(=O)NCC(OC)c1ccccc1C
COc1cc(C(=O)N(C)C[C@H](C)NC(=O)c2cc(F)ccc2N)n[nH]1
COc1cc(C(=O)N(C)[C@H](C)CC(=O)NC(C)Cc2cccs2)n[nH]1
COc1cc(C(=O)N(Cc2ccc(C)s2)CC23CCC(CC2)C3)sn1
COc1cc(C(=O)N2CC(OCc3nc(C)no3)C2)cc(OC)c1C
COc1cc(C(=O)N2CCCC(OC)(C(F)F)C2)nc2ccccc12
COc1cc(C(=O)N2C[C@@H](F)C[C@@H]2C(=O)N2CC(S(C)(=O)=O)C2)sn1
COc1cc(C(=O)NC2(C(=O)N3CC[C@@H]4[C@H]3C[C@H]4OC)CC2)ncn1
COc1cc(C(=O)NC2(c3ccc(Cl)cc3)COC2)cc(F)c1C#N
COc1cc(C(=O)NC2CC(NC(=O)C(C)N3CCOC3=O)C2)sn1
COc1cc(C(=O)NCC(C)(O)CNC(=O)[C@H]2C[C@@H]2C2CC2)ncn1
COc1cc(C(=O)NCC(C)(O)c2cc(C)oc2C)cc([N+](=O)[O-])c1
COc1cc(C(=O)NCC2=CCCN(C(=O)C(F)=CC3CC3)C2)sn1
COc1cc(C(=O)NCC2CC(CNC(=O)c3cnsn3)C2)ccn1
COc1cc(C(=O)NCCC(OC)C(C)C)ccc1OC1CCCC1
COc1cc(C(=O)NCCCC(C)NC(=O)Cc2ccno2)nn1C
COc1cc(C(=O)NC[C@H]2[C@@H](C(=O)NC(C)C(C)(C)C)C2(C)C)n[nH]1
COc1cc(C(=O)NCc2occc2C(=O)NCC(C)(C)SC)n[nH]1
COc1cc(C(=O)NNc2cc(C)c(C)nn2)c(C(F)F)cc1OC
COc1cc(C(=O)N[C@H](CC(C)C)C(=O)N2CCC(C)(O)CC2)n[nH]1
COc1cc(C(=O)Nc2c(C#N)oc3ccccc23)ccc1[N+](=O)[O-]
COc1cc(C(=O)O)nc(C(=O)N2CCc3ccc(F)cc3C2C)c1
COc1cc(C(=O)OCC(O)COCc2ccc(Cl)cc2)ccc1C
COc1cc(C(=O)OCCOCCC(=O)OC(C)(C)C)c(F)cc1Br
COc1cc(C(F)(F)F)ccc1CNC(=O)NNC(=O)NCC(F)F
COc1cc(C(F)F)ccc1CN1CCC(CCNS(N)(=O)=O)CC1
COc1cc(C)c(CN(C)C(=O)NCCc2cc(C)on2)cc1OC
COc1cc(C)c(CN2CC3(CCN(C)CC3)c3ccccc32)cn1
COc1cc(C)c2cc(C(=O)Nc3ccc(C)c(C4CC4)c3)[nH]c2c1
COc1cc(C)cc(C)c1C(=O)COC(=O)CN1CC(C)CS1(=O)=O
COc1cc(C)cc(CC(=O)NC[C@H](CF)NS(=O)(=O)CC2CC2)c1
COc1cc(C)cc(CN(CC2(Cl)CC2(F)F)C(=O)[C@H]2CC2(F)F)c1
COc1cc(C)cc(CN(Cc2cnn(C)c2)CC2CSCCS2)c1
COc1cc(C)ccc1C(=O)NCCN(C(=O)CC1CSC1)C1CC1
COc1cc(C)ccc1C(C(=O)NC(C)C)N1CCS(=N)(=O)C(C)C1
COc1cc(C)ccc1OCC(=O)NCc1ccc2ccn(C)c2c1
COc1cc(C)cnc1CN[C@H](CO)CCCNC(=O)OC(C)(C)C
COc1cc(C)ncc1C(N[C@H]1CC[C@H](CO)CC1)c1nnnn1C
COc1cc(C2CC2)ccc1NC(=O)N1CCC(C)(CS(C)(=O)=O)C1
COc1cc(C2CCN(C(=O)C(O)C(C)(C)C)C2)ccc1C(F)(F)F
COc1cc(C2CCN(C(=O)NC3COC(C)(C)C3)C2)cc(F)c1F
COc1cc(C=CC(=O)NCC(=O)NC2CNC2)cc(OC)c1OC
COc1cc(C=Cc2nc(-c3ccccc3)cs2)ccc1OCC#N
COc1cc(CC(=O)NNc2nc(C)ccc2[N+](=O)[O-])cnc1OC
COc1cc(CC(=O)Nc2ccc(N3CCCC(C)C3)c(Cl)c2)on1
COc1cc(CC(=O)OCCn2ccccc2=O)cc(OC)c1OC
COc1cc(CC(=O)Oc2c(C)cc(C)cc2Br)cc(OC)c1OC
COc1cc(CC(C)NC(=O)c2cc3ccc(C)cn3n2)ccc1O
COc1cc(CC(C)NCc2c[nH]c3cc(F)c(Cl)cc23)ccc1O
COc1cc(CCC(=O)NCCC(C)NS(=O)(=O)C2(C)CC2)ccn1
COc1cc(CCNC(=O)N(C)C2(c3cccnc3)CC2)cc(C)n1
COc1cc(CN(C)C(=O)c2cc(I)ccc2Cl)cc(OC)c1OC
COc1cc(CN(C)C)ccc1NC(=O)c1cnc2ccc(F)cn12
COc1cc(CN(C=O)[C@H](C)c2ccc3c(c2)CCCC3)c(F)cn1
COc1cc(CN(CC(C)OC(F)F)C(=O)[C@H]2CNC(=O)C2)ccn1
COc1cc(CN(CC(CO)C2CC2)C(=O)C(C)(O)C(F)(F)F)sn1
COc1cc(CN(CCC(C)(C)C)Cc2nccnc2C)cc(Cl)n1
COc1cc(CN(CCC2CC=CCC2)Cc2ncc(Cl)n2C)sn1
COc1cc(CN(CCC2CCSC2)C(=O)CCC(C)C)ccc1C
COc1cc(CN(Cc2cc(Br)[nH]n2)Cc2ccc(Cl)o2)c(Cl)cn1
COc1cc(CN(Cc2cc(C)c(C)cc2C)CC(F)C2CC2)sn1
COc1cc(CN(Cc2sc(C)nc2C)C[C@@H]2CCCC[C@H]2O)sn1
COc1cc(CN2[C@H](C)CC[C@@H]2C(=O)OC(C)(C)C)cc(OC)c1C
COc1cc(CNC(=O)C(=O)NCc2cc(C)cc(Cl)n2)ccc1F
COc1cc(CNC(=O)NCC2=NOC3OCCCC23)ccc1CO
COc1cc(CNC(=O)NCCOc2cc(Cl)ccc2F)ccc1Cl
COc1cc(CNC(=O)[C@H](C)n2cc(C3CCC3)nn2)c(Br)cc1C
COc1cc(CNC(=O)c2c(F)cc(F)c(O)c2F)cc(O)c1OC
COc1cc(CNC(=O)c2cc(O)ccn2)ccc1OCC(F)(F)F
COc1cc(CNC(=O)c2cnn3c2SCC3)ccc1OCC(N)=O